RVD-Hpα TFA

RVD-Hpα TFA is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. RVD-Hpα TFA increases intracellular Ca2+ levels in cells expressing CB1 receptors in vitro. RVD-Hpα TFA also high affinity CB2 positive allosteric modulator (Ki=50 nM).
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Reference:
HY-P1397A
Product Details
HY-P1397A

Data sheet

Size
Multiple sizes
Reactivity
Cannabinoid Receptor
Application
Neuroscience-Neuromodulation

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